Bioregulators

Epithalon

Also known as: Epitalon, Epithalone, AGAG

Clinical Trials
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Key Facts: Epithalon

Category
Bioregulators
FDA Status
Not FDA Approved
Clinical Status
Investigational - Primarily Russian research
Administration
Subcutaneous or intramuscular injection
Typical Dose
5-10 mg daily for 10-20 days
Frequency
Once daily in cycles
Evidence Level
Human Trials
Duration
10-20 day cycles
Also Known As
Epitalon, Epithalone, AGAG

What to Expect

A tetrapeptide studied for its effects on telomerase activation and potential anti-aging properties. Based on research by Professor Vladimir Khavinson.

Mechanism of Action

Epithalon stimulates telomerase production, potentially slowing or reversing telomere shortening. It may also regulate melatonin production by the pineal gland and has been shown to influence gene expression related to aging.

Research Summary

Russian studies show increased telomerase activity and extended lifespan in animal models. Human studies suggest improved sleep, reduced cortisol, and potential immune benefits. Research quality and Western replication remains limited.

Clinical Status:Investigational - Primarily Russian research
Trial Progress:Preclinical
Pre
I
II
III
IV
FDA

Dosing Information

Human Trials·Human studies conducted, not FDA approved

Typical Dosing

Community experience

Common Dose

5-10 mg daily for 10-20 days

Range

5-20 mg daily

Frequency

Once daily in cycles

Run in cycles of 10-20 days, then break for months. Targets telomerase activation. Usually done 1-2x per year.

Research Dosing

Scientific studies

Doses from research protocols

Doses from Studies

Duration

10-20 day cycles

Administration

Subcutaneous or intramuscular injection

Timing & Administration

Best Time to Take

Before bed

Once daily for 10-20 day cycles

Food Recommendation

With or without food

Why This Timing?

Epithalon supports telomere health and melatonin. Evening dosing aligns with natural repair processes during sleep.

Possible Side Effects

Not everyone experiences these effects. Individual responses vary based on dosage, duration, and personal factors.

  • Generally well-tolerated
  • Injection site reactions
  • Mild headache (transient)
  • Sleep disturbances
  • Risk of immunogenicity
  • Long-term safety not established

References

Related Peptides

Peptides commonly compared with Epithalon or used in similar applications.

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Educational Information Only

This information is provided for educational purposes only and is not intended as medical advice. Always consult with qualified healthcare providers before making any decisions about peptides or other substances. The protocols listed reflect doses observed in research studies, not recommendations.